 | | DRUG: Rizatriptan benzoate | |
| Entry |
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| Name |
Rizatriptan benzoate (JAN/USP);
Maxalt (TN) |
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| Product |
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| Generic |
RIZATRIPTAN (Bryant Ranch Prepack), RIZATRIPTAN (Macleods Pharmaceuticals Limited), RIZATRIPTAN BENZOATE (A-S Medication Solutions), RIZATRIPTAN BENZOATE (A-S Medication Solutions), RIZATRIPTAN BENZOATE (Ascend Laboratories), RIZATRIPTAN BENZOATE (Aurobindo Pharma Limited), RIZATRIPTAN BENZOATE (Aurobindo Pharma Limited), RIZATRIPTAN BENZOATE (Bionpharma Inc.,), RIZATRIPTAN BENZOATE (Breckenridge Pharmaceutical), RIZATRIPTAN BENZOATE (Breckenridge Pharmaceutical), RIZATRIPTAN BENZOATE (Bryant Ranch Prepack), RIZATRIPTAN BENZOATE (Bryant Ranch Prepack), RIZATRIPTAN BENZOATE (Bryant Ranch Prepack), RIZATRIPTAN BENZOATE (Bryant Ranch Prepack), RIZATRIPTAN BENZOATE (Cipla USA), RIZATRIPTAN BENZOATE (Creekwood Pharmaceuticals LLC), RIZATRIPTAN BENZOATE (DIRECT RX), RIZATRIPTAN BENZOATE (Direct Rx), RIZATRIPTAN BENZOATE (Direct_Rx), RIZATRIPTAN BENZOATE (Direct_Rx), RIZATRIPTAN BENZOATE (Glenmark Pharmaceuticals), RIZATRIPTAN BENZOATE (Glenmark Pharmaceuticals), RIZATRIPTAN BENZOATE (Golden State Medical Supply), RIZATRIPTAN BENZOATE (Golden State Medical Supply), RIZATRIPTAN BENZOATE (Macleods Pharmaceuticals Limited), RIZATRIPTAN BENZOATE (Mylan Pharmaceuticals), RIZATRIPTAN BENZOATE (NuCare Pharmaceuticals), RIZATRIPTAN BENZOATE (Panacea Biotec Limited), RIZATRIPTAN BENZOATE (Proficient Rx LP), RIZATRIPTAN BENZOATE (Proficient Rx LP), RIZATRIPTAN BENZOATE (Proficient Rx LP), RIZATRIPTAN BENZOATE (Proficient Rx LP), RIZATRIPTAN BENZOATE (Quality Care Products), RIZATRIPTAN BENZOATE (Quality Care Products), RIZATRIPTAN BENZOATE (RPK Pharmaceuticals), RIZATRIPTAN BENZOATE (RPK Pharmaceuticals), RIZATRIPTAN BENZOATE (Rising Pharma Holdings), RIZATRIPTAN BENZOATE (Rising Pharma Holdings), RIZATRIPTAN BENZOATE (Teva Pharmaceuticals USA), RIZATRIPTAN BENZOATE (Unichem Pharmaceuticals (USA)), RIZATRIPTAN BENZOATE (Unichem Pharmaceuticals (USA)), RIZATRIPTAN BENZOATE (direct rx), RIZATRIPTAN BENZOATE ODT (Direct Rx) |
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| Formula |
C15H19N5. C7H6O2
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| Exact mass |
391.2008
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| Mol weight |
391.4662
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| Structure |
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| Class |
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| Remark |
| Therapeutic category: | 2160 |
| Product (DG00838): | D00675<JP/US> |
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| Efficacy |
Antimigraine, Vasoconstrictor, Serotonin receptor agonist |
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| Comment |
Sumatriptan derivative
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| Target |
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| Pathway |
| hsa04080 | Neuroactive ligand-receptor interaction |
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| Interaction |
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| Structure map |
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| Brite |
Anatomical Therapeutic Chemical (ATC) classification [BR:br08303]
N NERVOUS SYSTEM
N02 ANALGESICS
N02C ANTIMIGRAINE PREPARATIONS
N02CC Selective serotonin (5HT1) agonists
N02CC04 Rizatriptan
D00675 Rizatriptan benzoate (JAN/USP) <JP/US>
USP drug classification [BR:br08302]
Antimigraine Agents
Serotonin (5-HT) Receptor Agonists
Rizatriptan
D00675 Rizatriptan benzoate (JAN/USP)
Therapeutic category of drugs in Japan [BR:br08301]
2 Agents affecting individual organs
21 Cardiovascular agents
216 Vasoconstrictors
2160 Vasoconstrictors
D00675 Rizatriptan benzoate (JAN/USP)
Drug groups [BR:br08330]
Analgesic
DG01484 5-HT1B-receptor agonist
DG00838 Rizatriptan
D00675 Rizatriptan benzoate
DG01485 5-HT1D-receptor agonist
DG00838 Rizatriptan
D00675 Rizatriptan benzoate
DG01518 5-HT1B/1D-receptor agonist
DG00838 Rizatriptan
D00675 Rizatriptan benzoate
DG01943 Triptan
DG00838 Rizatriptan
D00675 Rizatriptan benzoate
Target-based classification of drugs [BR:br08310]
G Protein-coupled receptors
Rhodopsin family
Serotonin
HTR1B
D00675 Rizatriptan benzoate (JAN/USP) <JP/US>
HTR1D
D00675 Rizatriptan benzoate (JAN/USP) <JP/US>
New drug approvals in Japan [br08318.html]
Drugs with new active ingredients
D00675
Drug groups [BR:br08330]
Analgesic
DG01484 5-HT1B-receptor agonist
DG00838 Rizatriptan
DG01485 5-HT1D-receptor agonist
DG00838 Rizatriptan
DG01518 5-HT1B/1D-receptor agonist
DG00838 Rizatriptan
DG01943 Triptan
DG00838 Rizatriptan
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| Other DBs |
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| KCF data |
ATOM 29
1 C8y C 30.1421 -18.0733
2 C8y C 30.1421 -19.4722
3 C8y C 31.4714 -17.6437
4 C8x C 28.9347 -17.3768
5 N4x N 31.4714 -19.9075
6 C8x C 28.9347 -20.1687
7 C8x C 32.2898 -18.7699
8 C8y C 27.7215 -18.0733
9 C8x C 27.7215 -19.4663
10 C1b C 26.5030 -17.3679
11 N4y N 25.3135 -18.0529
12 N5x N 25.3135 -19.4529
13 C8x C 23.9820 -17.6203
14 N5x N 23.1591 -18.7529
15 C8x C 23.9820 -19.8856
16 C1b C 31.4714 -16.2437
17 C1b C 32.7068 -15.5303
18 N1c N 33.9108 -16.2253
19 C1a C 35.0937 -15.5422
20 C1a C 33.9113 -17.6397
21 C8y C 39.2467 -17.9866
22 C8x C 38.0392 -18.6832
23 C8x C 40.4483 -18.6832
24 C6a C 39.2467 -16.5994
25 C8x C 38.0392 -20.0706
26 C8x C 40.4483 -20.0706
27 O6a O 40.4540 -15.9028
28 O6a O 38.0451 -15.9028
29 C8x C 39.2467 -20.7613
BOND 31
1 1 2 1
2 1 3 1
3 1 4 2
4 2 5 1
5 2 6 2
6 3 7 2
7 4 8 1
8 6 9 1
9 5 7 1
10 8 9 2
11 8 10 1
12 10 11 1
13 11 12 1
14 11 13 1
15 13 14 2
16 14 15 1
17 12 15 2
18 3 16 1
19 16 17 1
20 17 18 1
21 18 19 1
22 18 20 1
23 21 22 1
24 21 23 2
25 21 24 1
26 22 25 2
27 23 26 1
28 24 27 1
29 24 28 2
30 25 29 1
31 26 29 2
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